The Harmonizing Outcomes with Revascularization and Stents in Acute Myocardial Infarction Study (HORIZONS AMI)

Summary1

This large-scale, open-label, prospective, randomized trial of ST-segment elevation myocardial infarction (STEMI) patients undergoing a primary percutaneous coronary intervention (PCI) strategy, comparing Angiomax® (bivalirudin) vs unfractionated heparin (UFH) plus routine use of glycoprotein (GP) IIb/IIIa inhibitor monotherapy, at 30 days resulted in:1

– 24% reduction in the primary end point of net adverse clinical events (NACE)
– 41% reduction in the primary end point of major bleeding
– No difference in major adverse cardiovascular events (MACE)
– Reduced rate of both overall and cardiac mortality1

The multicenter, open-label, randomized trial of ST-segment elevation myocardial infarction (STEMI) patients undergoing a primary percutaneous coronary intervention (PCI) strategy. Of patients in the ANGIOMAX arm, the majority (93 percent) received ANGIOMAX monotherapy. At one year, results showed that, compared with the control treatment, ANGIOMAX:

– Reduced the incidence of cardiac-related death by 43 percent (2.1% vs. 3.8%, HR 0.57 [95% CI 0.38-0.84]; P=0.005)
– Reduced all-cause death by 31 percent (3.4% vs. 4.8%, HR 0.70 [95% CI 0.50-0.97]; P=0.029)
– Reduced the incidence of net adverse clinical events, a composite of major adverse cardiac events or major bleeding, by 16 percent (15.7% vs. 18.3%, HR 0.84 [95% CI 0.71-0.98]; P=0.03)
– Reduced rates of major bleeding by 39 percent (5.8% vs. 9.2%, HR 0.61 [95% CI 0.48-0.78]); P<0.0001)
– Demonstrated no difference in rates of major adverse cardiac events (11.9% vs. 11.9%, HR 1.00 [95% CI 0.83-1.21]; P=0.98)

Trial Design

HORIZONS AMI findings support ANGIOMAX use in STEMI patients undergoing primary PCI

* ANGIOMAX monotherapy included "provisional" GP IIb/IIIa inhibitor.
The safety and effectiveness of ANGIOMAX have not been established in patients with acute coronary syndromes (ACS) who are not undergoing PCI.4

Inclusion Criteria1

Exclusion Criteria

Clinical Endpoints1

Primary Endpoints (at 30 days)1

HORIZONS-AMI 30-Day End Point1

TVR=target vessel revascularization

Baseline Characteristics1

Bivalirudin*
(n=1,800)
UFH + GP IIb/IIIa
(n=1,802)
Age, years [range] 59.8 [26.0-92.3] 60.7 [21.6–91.6]
Male 77.1% 76.1%
Diabetes 15.6% 17.3%
HTN 51.8% 55.2%
Hyperlipidemia 43.4% 42.7%
Current smoking 47.2% 45.0%
Prior MI 10.4% 11.4%
Prior PCI 10.5% 11.0%
Prior CABG 3.3% 2.6%
Weight, kg [range] 80 [71–90.3] 80 [71–90]
Chest pain – ED, hours [range] 2.2 [1.3–4.0] 2.1 [1.3–3.9]
Killip class 2-4 8.5% 8.5%
LVEF, % [range] 50 [45–60] 50 [41–59]

* In HORIZONS AMI: 93% of ANGIOMAX patients received ANGIOMAX monotherapy1

ANGIOMAX significantly reduced NACE* and major bleeding with no difference in MACEat 30 days in HORIZONS AMI1 these results were maintained at 1 year5

* NACE=MACE or major bleeding.1
MACE=major adverse cardiovascular events: all-cause death, reinfarction, ischemic target vessel revascularization, or stroke.1
IN HORIZONS AMI, 93% of ANGIOMAX patients received ANGIOMAX monotherapy, without provisional GP IIb/IIIa inhibitor.1
§ Data from Kaplan-Meier analyses based on log-rank estimates.
|| Non-CABG.

ANGIOMAX resulted in lower rates of overall and cardiac mortality at 30-days1 and 1-year in HORIZONS AMI 5

* IN HORIZONS AMI, 93% of ANGIOMAX patients received ANGIOMAX monotherapy, without provisional GP IIb/IIIa inhibitor.1
Data from Kaplan-Meier analyses based on log-rank estimates.
Please see important safety information and bleeding definitions.

Similar Rates of Stent Thrombosis Between Treatment Groups at 30 Days and 1 Year

* Protocol definition of stent thrombosis, CEC adjudicated.
In HORIZONS AMI, 93% of bivalirudin patients received monotherapy, without provisional GP IIb/IIIa inhibitor.
ARC=Academic Research Consortium; CEC=clinical events committee..

In HORIZONS AMI, more deaths were attributed to 30-day major bleeding—association between 30-day events and 30-day mortality in HORIZONS AMI1,7

More deaths were attributable to major bleeding than stent thrombosis

* Time-updated covariate-adjusted Cox model.
Attributable deaths = N deaths among patients with the time updated event (attribute) X (adj. HR – 1)/adjusted HR.
6.5% of 93 total deaths.
29.0% of 93 total deaths.

Reduction in 1-Year Overall Mortality demonstrated with ANGIOMAX, Regardless of Stent Type5

* In HORIZONS AMI, 93% of bivalirudin patients received monotherapy, without provisional GP IIb/IIIa inhibitor.

Safety Considerations
ANGIOMAX with provisional use of glycoprotein IIb/IIIa inhibitor is indicated for use as an anticoagulant in patients undergoing percutaneous coronary intervention (PCI), and in patients with or at risk for heparin-induced thrombocytopenia and thrombosis syndrome (HIT/HITTS) undergoing PCI. ANGIOMAX is intended for use with aspirin and has been studied only in patients receiving concomitant aspirin. ANGIOMAX is contraindicated in patients with active major bleeding or hypersensitivity to ANGIOMAX or its components. The most common (≥10%) adverse events for ANGIOMAX were back pain, pain, nausea, headache, and hypotension. An unexplained fall in blood pressure or hematocrit, or any unexplained symptom, should lead to serious consideration of a hemorrhagic event and cessation of ANGIOMAX administration. Please see complete prescribing information.

1Stone GW, Witzenbichler B, Guagliumi G, et al; for the HORIZONS AMI trial investigators. Bivalirudin during primary PCI in acute myocardial infarction. N Engl J Med. 2008;358:2218-2230.

2Lincoff AM, Bittl JA, Harrington RA, et al. Bivalirudin and provisional glycoprotein IIb/IIIa blockade compared with heparin and planned glycoprotein IIb/IIIa blockade during percutaneous coronary intervention: REPLACE-2 randomized trial. JAMA. 2003;289:853-863.

3Stone GW, McLaurin BT, Cox DA, et al; for the ACUITY Investigators. Bivalirudin for patients with acute coronary syndromes. N Engl J Med. 2006;355:2203-2216.

4ANGIOMAX Prescribing Information. The Medicines Company; Parsippany, NJ, December 6, 2005

5Mehran R; HORIZONS-AMI Trial Investigators. A prospective, randomized comparison of bivalirudin vs. heparin plus glycoprotein IIb/IIIa inhibitors during primary angioplasty in acute myocardial infarction—one year results [oral presentation]. Presented at: Transcatheter Cardiovascular Therapeutics (TCT); October 12-17, 2008;
Washington, DC.

6Mauri L, Hsieh WH, Massaro JM, Ho KKL, D’Agostino R, Cutlip DE. Stent thrombosis in randomized clinical trials of drug-eluting stents. N Engl J Med. 2007;356:1020-1029.

7Data on file. The Cardiovascular Research Foundation, New York, NY.

© 2008 The Medicines Company
Acute Care Hospital Products
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